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分类: Total Synthesis

Total synthesis of (±)-3-demethoxyerythratidinone via Tf2O-promoted cascade reaction of enaminone

2025-10-16 by admin

Mingliang Lou, Xiaolei Liu, Shoule Han, Songlin Bai and …

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Triflic Anhydride Promoted Decarboxylative Functionalization of α-Amino Acids

2025-10-16 by admin

Mingyue Yuan, Mingliang Lou, Gen Li and Xiangbing Qi Th …

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Total Synthesis of Tetracyclic Spirooxindole Alkaloids via a Double Oxidative Rearrangement/Cyclization Cascade

2025-10-16 by admin

Xin Wang, Mengjiao Zhang, Xiaolei Liu, Mingliang Lou, G …

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A brief overview of classical natural product drug synthesis and bioactivity

2025-10-16 by admin

Gen Li, Mingliang Lou and Xiangbing Qi Traditional medi …

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Total Synthesis of Tetrodotoxin and 9-epiTetrodotoxin

2025-10-16 by admin

Peihao chen ,Jing Wang ,Yan Wang ,Yuze Sun ,Songlin Bai …

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Bioinspired Formal Synthesis of Pancracine via Selective Hydrogenation of Indole Derivative

2025-10-16 by admin

Shoule Han, Mingliang Lou Xiangbing Qi* In drug develop …

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Oxidative Coupling Approach to Sarpagine Alkaloids: Total Synthesis of (−)-Trinervine, Vellosimine, (+)-Normacusine B, and (−)-Alstomutinine C

2023-05-12 by admin

Ye Zhang, Lei Zhang, Xiangbing Qi* Sarpagine alkaloids …

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Asymmetric Total Syntheses of Strychnos Alkaloids via Selective Fischer Indolization

2022-10-08 by admin

Xiaolei Liu, Mingliang Lou, Songlin Bai, Guoxin Sun,* a …

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Flavin-Dependent Monooxygenase-Mediated 1,2-Oxazine Construction via Meisenheimer Rearrangement in the Biosynthesis of Paeciloxazine

2022-02-28 by admin

Daojiang Yan, Kunya Wang, Songlin Bai, Bingyu Liu, Jian …

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Total Synthesis of (-)-Alstofolinine A through a Furan Oxidation/ Rearrangement and Indole Nucleophilic Cyclization Cascade

2021-12-10 by admin

Lei Zhang, Ye Zhang, Wenting Li, and Xiangbing Qi*     …

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News

  • Radical Ring Expansion Catalyzed by an α-Ketoglutarate-Dependent Dioxygenase in the Biosynthesis of Tropolones
  • Cp*Ir(III)-Catalyzed Asymmetric Tandem Intramolecular Aziridination/Aza-Semipinacol Rearrangement of Alkenyl 1,4,2-Dioxazol-5-one
  • Structure-Based Optimization of TBK1 Inhibitors
  • Total synthesis of (±)-3-demethoxyerythratidinone via Tf2O-promoted cascade reaction of enaminone
  • Dissecting caspase-2-mediated cell death: from intrinsic PIDDosome activation to chemical modulation
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