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分类: Medicinal chemistry

Estrogen-Related Hormones Induce Apoptosis by Stabilizing Schlafen-12 Protein Turnover

2021-12-13 by admin

Dianrong Li, Jie Chen, Youwei Ai, Xiaoqiong Gu, Li Li, …

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Staurosporine targets the Hippo pathway to inhibit cell growth

2021-12-13 by admin

Xueyan Ma, Peixue Li, Peihao Chen, Jinhui Li, Hongling …

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A general strategy for synthesis of cyclophane-braced peptide macrocycles via palladium-catalysed intramolecular sp 3 C-H arylation

2021-12-13 by admin

Xuekai Zhang, Gang Lu, Meng Sun, Madhu Mahankali, Yanfe …

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A Novel Inhibitor of Pyruvate Dehydrogenase Kinase Stimulates Myocardial Carbohydrate Oxidation in Diet-Induced Obesity

2021-12-10 by admin

Cheng-Yang Wu, Santhosh Satapati, Wenjun Gui, Richard M …

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A hybridization-chain-reaction-based method for amplifying immunosignals

2021-12-13 by admin

Rui Lin, Qiru Feng, Peng Li, Ping Zhou, Ruiyu Wang, Zhe …

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Targeting hepatic pyruvate dehydrogenase kinases restores insulin signaling and mitigates ChREBP-mediated lipogenesis in diet-induced obese mice

2021-04-28 by admin

Cheng-Yang Wu, Shih-Chia Tso, Jacinta L. Chuang, Wen-Ju …

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a hybridiza-tionchain-reaction-based method for amplifying immunosignals

2021-04-28 by admin

Rui Lin, Qiru Feng, Peng Li, Ping Zhou, Ruiyu Wang, Zhe …

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In Silico Identification of a Novel Hinge-Binding Scaffold for Kinase Inhibitor Discovery

2021-04-28 by admin

Yanli Wang, Yuze Sun, Ran Cao, Dan Liu, Yuting Xie, Li …

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Development of Dihydroxyphenyl Sulfonylisoindoline Derivatives as Liver-Targeting Pyruvate Dehydrogenase Kinase Inhibitors

2021-04-28 by admin

Shih-Chia Tso, Mingliang Lou, Cheng-Yang Wu, Wen-Jun Gu …

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Reciprocal Regulation between the Circadian Clock and Hypoxia Signaling at the Genome Level in Mammals

2021-04-28 by admin

Yaling Wu, Dingbin Tang, Na Liu, Wei Xiong, Huanwei Hua …

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News

  • Flavin-Dependent Monooxygenase-Mediated 1,2-Oxazine Construction via Meisenheimer Rearrangement in the Biosynthesis of Paeciloxazine
  • Expeditious and Efficient ortho-Selective Trifluoromethane-sulfonylation of Arylhydroxylamines
  • An improved auxin-inducible degron system for fission yeast
  • Structure of PDE3A–SLFN12 complex and structure-based design for a potent apoptosis inducer of tumor cells
  • 5-IP7: a GPCR messenger mediating muscarinic control of synaptotagmin-dependent insulin exocytosis and glucose homeostasis
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