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分类: Publications

A general strategy for synthesis of cyclophane-braced peptide macrocycles via palladium-catalysed intramolecular sp 3 C-H arylation

2021-12-13 by admin

Xuekai Zhang, Gang Lu, Meng Sun, Madhu Mahankali, Yanfe …

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A Novel Inhibitor of Pyruvate Dehydrogenase Kinase Stimulates Myocardial Carbohydrate Oxidation in Diet-Induced Obesity

2021-12-10 by admin

Cheng-Yang Wu, Santhosh Satapati, Wenjun Gui, Richard M …

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Development of the Vinylogous Pictet–Spengler Cyclization and Total Synthesis of (±)-Lundurine A

2021-12-10 by admin

Aaron Nash, Xiangbing Qi, Pradip Maity, Kyle Owens, and …

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A hybridization-chain-reaction-based method for amplifying immunosignals

2021-12-13 by admin

Rui Lin, Qiru Feng, Peng Li, Ping Zhou, Ruiyu Wang, Zhe …

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A general strategy for synthesis of cyclophanebraced peptide macrocycles via palladiumcatalysed intramolecular sp3 C−H arylation

2021-04-28 by admin

Xuekai Zhang, Gang Lu, Meng Sun, Madhu Mahankali, Yanfe …

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Targeting hepatic pyruvate dehydrogenase kinases restores insulin signaling and mitigates ChREBP-mediated lipogenesis in diet-induced obese mice

2021-04-28 by admin

Cheng-Yang Wu, Shih-Chia Tso, Jacinta L. Chuang, Wen-Ju …

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a hybridiza-tionchain-reaction-based method for amplifying immunosignals

2021-04-28 by admin

Rui Lin, Qiru Feng, Peng Li, Ping Zhou, Ruiyu Wang, Zhe …

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In Silico Identification of a Novel Hinge-Binding Scaffold for Kinase Inhibitor Discovery

2021-04-28 by admin

Yanli Wang, Yuze Sun, Ran Cao, Dan Liu, Yuting Xie, Li …

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Development of Dihydroxyphenyl Sulfonylisoindoline Derivatives as Liver-Targeting Pyruvate Dehydrogenase Kinase Inhibitors

2021-04-28 by admin

Shih-Chia Tso, Mingliang Lou, Cheng-Yang Wu, Wen-Jun Gu …

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Reciprocal Regulation between the Circadian Clock and Hypoxia Signaling at the Genome Level in Mammals

2021-04-28 by admin

Yaling Wu, Dingbin Tang, Na Liu, Wei Xiong, Huanwei Hua …

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News

  • Radical Ring Expansion Catalyzed by an α-Ketoglutarate-Dependent Dioxygenase in the Biosynthesis of Tropolones
  • Cp*Ir(III)-Catalyzed Asymmetric Tandem Intramolecular Aziridination/Aza-Semipinacol Rearrangement of Alkenyl 1,4,2-Dioxazol-5-one
  • Structure-Based Optimization of TBK1 Inhibitors
  • Total synthesis of (±)-3-demethoxyerythratidinone via Tf2O-promoted cascade reaction of enaminone
  • Dissecting caspase-2-mediated cell death: from intrinsic PIDDosome activation to chemical modulation
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