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Discovery of a molecular glue promoting CDK12-DDB1 interaction to trigger cyclin K degradation

2021-12-13 by admin

Lu Lv, Peihao Chen, Longzhi Cao, Yamei Li, Zhi Zeng, Yu …

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An alkaloid initiates phosphodiesterase 3A–schlafen 12 dependent apoptosis without affecting the phosphodiesterase activity

2021-12-13 by admin

Youwei Ai, Haibing He, Peihao Chen, Bo Yan, Wenbin Zhan …

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Visible-light-induced Nickel-catalyzed Chemoselective Cross-coupling of gem-Borazirconocene Alkanes with Aryl Halides

2021-12-10 by admin

Chao Yang, Yadong Gao, Songlin Bai, Chao Jiang,* and Xi …

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Direct Synthesis of Annulated Indoles through Palladium-Catalyzed Double Alkylations

2021-12-10 by admin

Yadong Gao, Jianhua Li, Songlin Bai, Daoquan Tu, Zhiwen …

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Chemical perturbations reveal that RUVBL2 regulates the circadian phase in mammals

2021-12-13 by admin

Dapeng Ju, Wei Zhang, Jiawei Yan, Haijiao Zhao, Wei Li, …

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Visible-Light-Induced Nickel-Catalyzed Cross-Coupling with Alkylzirconocenes from Unactivated Alkenes

2021-12-10 by admin

Yadong Gao, Chao Yang, Songlin Bai, Xiaolei Liu, Qingcu …

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A thiazole-derived oridonin analog exhibits antitumor activity by directly and allosterically inhibiting STAT3

2021-12-10 by admin

Xiaofei Shen 1, Lin Zhao 1, Peihao Chen, Yanqiu Gong, D …

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Estrogen-Related Hormones Induce Apoptosis by Stabilizing Schlafen-12 Protein Turnover

2021-12-13 by admin

Dianrong Li, Jie Chen, Youwei Ai, Xiaoqiong Gu, Li Li, …

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Total Synthesis of (-)-Alstofolinine A through a Furan Oxidation/ Rearrangement and Indole Nucleophilic Cyclization Cascade

2021-12-10 by admin

Lei Zhang, Ye Zhang, Wenting Li, and Xiangbing Qi*     …

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Staurosporine targets the Hippo pathway to inhibit cell growth

2021-12-13 by admin

Xueyan Ma, Peixue Li, Peihao Chen, Jinhui Li, Hongling …

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News

  • Unlocking the secrets to human NTCP structure
  • BAFinder: A software for unknown bile acid identification using accurate mass LC-MS/MS in positive and negative modes
  • Asymmetric Total Syntheses of Strychnos Alkaloids via Selective Fischer Indolization
  • Flavin-Dependent Monooxygenase-Mediated 1,2-Oxazine Construction via Meisenheimer Rearrangement in the Biosynthesis of Paeciloxazine
  • Expeditious and Efficient ortho-Selective Trifluoromethane-sulfonylation of Arylhydroxylamines
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